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PNU-120596 and 3-(2,4-dimethoxybenzylidene) Anabaseine (GTS-21) (both nAchRa7 agonists) and Methyllycaconitine (anAchRa7 antagonist), are Highly Effective Drugs in Therapy of Ulcerative Colitis (UC) and
Crohn's Disease
(CD)
C10382: Breakthrough Therapeutic for Inflammatory Bowel Diseases (IBD)Novelty: This technology identifies a nicotinic acetylcholine receptor isoform (nAChR7) that has a prevalent role in affecting Inflammatory Bowel Disease (IBD), as well as several agonist/antagonists to nAChR7, that are highly effective in both the prevention and therapy of ulcerative...
Published: 3/13/2025
|
Inventor(s):
Philip Alex
,
Michael Centola
,
Xuhang Li
Keywords(s):
Chronic Inflammatory Diseases
,
Combination
,
Crohn's disease
,
Crohn's Disease
,
Disease Indication
,
Gastrointestinal Disorders
,
Inflammatory Bowel Disease
,
Inflammatory Bowel Disease (IBD)
,
Natural compounds
,
Non-novel
,
Off-the-shelf
,
Predicted Novelty
,
Small Molecules
,
Targeted Therapy/Targeted Therapy
,
Therapeutic Matter
,
Therapeutic Substance
,
Therapeutics
,
Therapy Type
,
Ulcerative Colitis
,
Ulcerative Colitis (UC)
Category(s):
Clinical and Disease Specializations
,
Clinical and Disease Specializations > Gastroenterology >
Crohn's Disease
,
Clinical and Disease Specializations > Gastroenterology > Inflammatory Bowel Disease
,
Clinical and Disease Specializations > Gastroenterology > Ulcerative Colitis
,
Clinical and Disease Specializations > Inflammation > Chronic Inflammatory Diseases
,
Clinical and Disease Specializations > Rare Diseases
,
Technology Classifications > Therapeutic Modalities > Small Molecules
,
Technology Classifications > Therapeutic Modalities > Targets
,
Clinical and Disease Specializations > Gastroenterology
,
Clinical and Disease Specializations > Inflammation
,
Technology Classifications > Therapeutic Modalities
PNU-120596 and 3-(2,4-dimethoxybenzylidene) Anabaseine (GTS-21) (both nAchRa7 agonists) and Methyllycaconitine (anAchRa7 antagonist), are Highly Effective Drugs in Therapy of Ulcerative Colitis (UC) and
Crohn's Disease
(CD)
C10382: Breakthrough Therapeutic for Inflammatory Bowel Diseases (IBD)Novelty: This technology identifies a nicotinic acetylcholine receptor isoform (nAChR7) that has a prevalent role in affecting Inflammatory Bowel Disease (IBD), as well as several agonist/antagonists to nAChR7, that are highly effective in both the prevention and therapy of ulcerative...
Published: 3/13/2025
|
Inventor(s):
Philip Alex
,
Michael Centola
,
Xuhang Li
Keywords(s):
Chronic Inflammatory Diseases
,
Combination
,
Crohn's disease
,
Crohn's Disease
,
Disease Indication
,
Gastrointestinal Disorders
,
Inflammatory Bowel Disease
,
Inflammatory Bowel Disease (IBD)
,
Natural compounds
,
Non-novel
,
Off-the-shelf
,
Predicted Novelty
,
Small Molecules
,
Targeted Therapy/Targeted Therapy
,
Therapeutic Matter
,
Therapeutic Substance
,
Therapeutics
,
Therapy Type
,
Ulcerative Colitis
,
Ulcerative Colitis (UC)
Category(s):
Clinical and Disease Specializations
,
Clinical and Disease Specializations > Gastroenterology >
Crohn's Disease
,
Clinical and Disease Specializations > Gastroenterology > Inflammatory Bowel Disease
,
Clinical and Disease Specializations > Gastroenterology > Ulcerative Colitis
,
Clinical and Disease Specializations > Inflammation > Chronic Inflammatory Diseases
,
Clinical and Disease Specializations > Rare Diseases
,
Technology Classifications > Therapeutic Modalities > Small Molecules
,
Technology Classifications > Therapeutic Modalities > Targets
,
Clinical and Disease Specializations > Gastroenterology
,
Clinical and Disease Specializations > Inflammation
,
Technology Classifications > Therapeutic Modalities
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